Downstream synthetic route of 51149-08-7

51149-08-7 3,6-Dichloropyridazine-4-carboxylic acid 433804, apyridazine compound, is more and more widely used in various fields.

With the rapid development and complex challenges of chemical substances, new drug synthesis pathways are usually the most effective.51149-08-7,3,6-Dichloropyridazine-4-carboxylic acid,as a common compound, the synthetic route is as follows.

51149-08-7, Example 5( 6-Chloro-1 H -indol-3-yl)[ 6-chloro-[3-( 4-.fluorobenzyl)amino ]pyridazin-4-yl]methanone 3,6-Dichloropyridazine-4-carbonyl chloride. 3,6-Dichloropyridazine-4-carboxylic acid (Aldrich; 1.13 g, 5.86 mmol) in toluene (20 mL) containing 2 drops of DMF was treated with neat SOCI2 (4 mL). The mixture heated to reflux for 3h and then allowed to cool. The resulting red-orange mixture was decanted and cone, in vacuo. The residue was redis solved in toluene and cone to give 1.22 g of the product.

51149-08-7 3,6-Dichloropyridazine-4-carboxylic acid 433804, apyridazine compound, is more and more widely used in various fields.

Reference£º
Patent; THE REGENTS OF THE UNIVERSITY OF CALIFORNIA; HOGENKAMP, Derk; WO2013/169907; (2013); A1;,
Pyridazine – Wikipedia
Pyridazine | C4H4N2 – PubChem